Mocetinostat


Induces hyperacetylation of histones, induces expression of the tumor suppressor p21WAF1 and inhibits proliferation of human cancer cells. Displays antifibrotic effects in ischemic heart failure. Attenuates the development of hypersensitivity in models of neuropathic pain. Active in vivo.

Amount: 5mg

Physical Properties: Off-white crystalline powder

MW=396.4 C₂₃H₂₀N₆O

Analysis: >98% (HPLC); NMR (Conforms)

Solubilization: May be dissolved in DMSO (25 mg/ml)

Storage: Store desiccated at ambient temperature for up to 2 years. Store solutions at -20°C for up to 2 months.