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CPTH2

Part Number:EI-HAT-003
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CPTH2



Cyclopentylidene-[4-(4’-chlorophenyl)thiazol-2-yl]hydrazone, CPTH2 is a selective inhibitor of the histone acetyltransferase Gcn5P both in vitro and in vivo (IC50 = 0.800 mM). In vitro, the HAT inhibitory activity of CPTH2 was caused via bridge-interaction with histone H3. In vivo it decreased acetylation of bulk histone H3 at the H3-AcK14 site.

Amount: 5mg

Physical Properties: White powder

MW=291.8 C14H14ClN3S

Analysis: >98% (TLC); NMR (Conforms)

Solubilization: May be dissolved in DMSO (>25 mg/ml)

Storage: Store desiccated as supplied at -20°C for up to 2 years. Store solutions at -20°C for up to one month.