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Your Price:$85.00
In Stock.
Part Number:EI-HAT-003

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Cyclopentylidene-[4-(4’-chlorophenyl)thiazol-2-yl]hydrazone, CPTH2 is a selective inhibitor of the histone acetyltransferase Gcn5P both in vitro and in vivo (IC50 = 0.800 mM).  In vitro, the HAT inhibitory activity of CPTH2 was caused via bridge-interaction with histone H3. In vivo it decreased acetylation of bulk histone H3 at the H3-AcK14 site.

Amount: 5mg

Physical Properties:  White powder 

MW=291.8          C14H14ClN3S

Analysis:  >98% (TLC); NMR (Conforms)

Solubilization: May be dissolved in DMSO (>25 mg/ml)

Storage:  Store desiccated as supplied at -20°C for up to 2 years. Store solutions at -20°C for up to one month.

With the largest functional kinase activity assay panel in the industry, RBC provides kinase, epigenetic, and other profiling services to over 590 companies worldwide. RBC specializes in custom assay conditions, high quality reproducible data, and outstanding service.

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